Proteros Biostructures Newsletter: January 2025

Proteros Biostructures Newsletter: January 2025

Excellence is our main asset

Excellence in project execution is fundamental - we deliver what we promise. We reach the milestones, meet timelines and agreed budgets. Our expertise warrants the design of scientifically relevant experiments that ultimately reach the RIGHT outcomes.

Learn more about our scientific excellence


Biological characterization of AB-343, a novel and potent SARS-CoV-2-Mpro inhibitor with pan-coronavirus activity

PROTEROS and Arbutus Biopharma co-publish study on the identification of Macrocyclic novel noncovalent inhibitors of SARS-CoV-2 Mpro.?

The recent global COVID-19 pandemic has highlighted treatments for coronavirus infections. The main protease (Mpro) has been an important target for the development of SARS-CoV-2 direct-acting antivirals. Proteros supported Arbutus with the identification and verification of these novel inhibitors in this project by designing and accurately producing the necessary purified Mpro protein and associated off-target proteins for proteolytic inhibition assays as well as ultra-pure protein for x-ray crystallography experiments. Assay ready proteins were utilized to identify IC50 values of various Macrocycles, along with kinetic binding measurements performed via in-house SPR. Finally, Co-crystal structures were delivered to confirm the binding mode of top performing Macrocycles.

See the full article at the link below to learn more and inquire with us at PROTEROS to discuss your program needs.

Read Publication Here


New Gallery Structures, Proteins and Assays now available at PROTEROS!

New Gallery Structures for Crystallography Include:?

  • RIPK-3, Murin
  • IL17A, Human
  • Androgen Receptor, Human
  • Thyroid Hormone Receptor Beta, Human
  • Trek-2 Channel, Human
  • HSD17B13, Human

New Gallery Structures for Cryo-EM Include:?

  • STTR2: Active
  • A2AR Active / Inactive State GPCR?
  • Dopamine Receptor?
  • GPR120 Active?
  • GPR61 Inactive?
  • Human Voltage Gated Potassium KV1.3 Channel?
  • Cyclin H-CDK7-Mat1 Complex?
  • DDB1: DCAF PROTAC and glue (Multiple Complexes)?
  • DDB1: CRBN PROTAC and glue (Multiple Complexes)?
  • 20S Proteosome

See the full list of available "off-the-shelf" proteins, structures and assays that are available to help kick-start your drug discovery program.

See Gallery List


Our Services

DISCOVERY SOLUTIONS

We serve as our client's innovative catalyst, leveraging our cutting-edge technology platform and expert knowledge to drive novel solutions in drug discovery.

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X-RAY CRYSTALLOGRAPHY

Elucidation of even the most complex structures through the preparation of the RIGHT protein.

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ASSAYS, BIOPHYSICS & SCREENING

Our diverse range of services includes both pre-established and tailor-made assay development solutions designed specifically for profiling and screening applications.

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BIOLOGICS

Your "one-stop-shop" solution for complex biologics / antigen purification with biochemical, biophysical and structural characterization.

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CRYO-EM

Cutting edge Cryo-EM technology platform to deliver the RIGHT challenging proteins and complexes.

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PROTEIN SCIENCES

At the heart of everything we do is the RIGHT protein for the right experiment. We ensure all proteins have the necessary unique characteristics to ensure your programs success.

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PROVEN TRACK RECORD AT PROTEROS

Proven track record with 200+ pharma and biotech partners in US, Europe and Japan. Serving most of the world's 20 largest pharma companies.

Providing discovery support to hundreds of big, small, and virtual biotechs.

6,000+ Structures elucidated

10,000+ Projects completed

300+ Peer-reviewed publications


Cutting Edge Facilities to Foster Excellence

Located in the thriving Martinsried / Munich - Biotech Cluster in Germany, our cutting-edge facility has been meticulously designed to cater to our specific service execution demands. Each specialized area, including Structural Biology, Cryo-EM, Protein Sciences, Biologics, Biophysics and Screening, has dedicated floors and lab rooms. We have created an environment where all these disciplines coexist under one roof, fostering the seamless collaboration and synergistic interaction necessary for the success of Discovery Solutions and multi-disciplinary projects.

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Copyright ? 2025 Proteros Biostructures GmbH

Mailing address:

EUROPE

Tel: +49 (0)89/700761-0 Fax: +49 (0)89-700761-115 Email: [email protected]

Headquarters: Proteros biostructures GmbH Bunsenstrasse 7a, D-82152 Martinsried Germany Get directions

NORTH AMERICA

Tel: +1-213-924-1483 Email: [email protected]

Headquarters: Proteros USA Inc. One Broadway, 14th Floor, Cambridge, MA 02142 United States Get directions

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