Med. Chem. Res. 2023, Vol 32, Iss 6

Med. Chem. Res. 2023, Vol 32, Iss 6

Medicinal Chemistry Research (Med Chem Res, MCR) Medicinal Chemistry Research (Med Chem Res, MCR)

Medicinal Chemistry Research (Med Chem Res, MCR)

An International Journal Promoting Bioactive Compounds, published by Springer Science+Business Media, Springer Nature

发布日期: 2023年6月10日
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Medicinal Chemistry Research | 2023 | ?Volume 32, Issue 6, ?is now available online.

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In this issue

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Review Article

Exploring the potential of chromone scaffold compounds in cancer therapy: targeting key kinase pathways

Rajibul Islam, Md. Selim Hossain, Phooi Yan Mock, Sze Wei Leong, Kok Wai Lam

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Review Article

An update on the discovery and development of reversible covalent inhibitors

Faridoon, Raymond Ng, Guiping Zhang, Jie Jack Li

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Review Article

Promising Schiff bases in antiviral drug design and discovery

Shikha Kaushik, Sarvesh Kumar Paliwal, Malliga R. Iyer, Vaishali M. Patil

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Original Research

Design, synthesis, biochemical and in silico characterization of novel naphthalene-thiourea conjugates as potential and selective inhibitors of alkaline phosphatase

Aamer Saeed, Saba Ashraf, Mubashir Aziz, Pervaiz Ali Channar, Syeda Abida Ejaz, Ammara Fayyaz, Qamar Abbas, Fatmah Ali Alasmary, Abdulnasser Mahmoud Karami, Arfa Tehzeeb, Amara Mumtaz, Hesham R. El-Seedi

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Original Research

Design, synthesis, and anti-aging effect evaluation of urolithin B and its amide derivatives on nematode Caenorhabditis elegans

Xi Chen, Xiaoqing Feng, Xiangming Kong, Hecheng Wang, Tianwen Liu, Long Tang, Ziheng Zhuang

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Original Research

Design & synthesis of hybrid pharmacophore of β-lactam, 1,8-naphthyridine, and secondary amines; Discover their in vitro antimicrobial, anticancer properties & DFT and ADMET prediction studies

Keyur M. Pandya, Satyanarayana Battula, K. A. Aravinda Kumar, Rajesh J. Patel, Navin B. Patel

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Original Research

Development of phosphoinositide 3-kinase delta (PI3Kδ) inhibitors as potential anticancer agents through the generation of ligand-based pharmacophores and biological screening

Mahmoud A. Al-Sha’er, Mutasem Taha, Mahmoud A. Alelaimat

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Original Research

Synthesis and evaluation of novel 3, 4-dihydropyrimidin-2(1H)- thione based pongamol conjugates as antibacterial agents

Anjaneyulu Eanti, Rajesh Gujju, Sunil Misra, Siddaiah Vidavalur, Sanjit Kanjilal

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Original Research

Design, synthesis and biological evaluation of aminopyrimidine derivatives bearing dihydroquinoxalinone as novel EGFRL858R/T790M kinase inhibitors against non-small-cell lung cancer

Liping Fu, Yu Cao, Jingbai Chen, Ruoyu He, Yanmei Zhao, Yaping Zhao, Jianjun Xi, Rangxiao Zhuang, Chongmei Tian

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Original Research

Design, synthesis, molecular docking study and molecular dynamics simulation of new coumarin-pyrimidine hybrid compounds having anticancer and antidiabetic activity

Duong Ngoc Toan, Nguyen Dinh Thanh, Mai Xuan Truong, Dinh Thuy Van, Nguyen Ngoc Thanh

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Original Research

Antiproliferative activity of secondary metabolites isolated from Humboldtia unijuga Bedd.

Reshma Vijayakumari Raveendran Nair, Ajikumaran Nair Sadasivan Nair, Anil John Johnson, Ananthakrishnan Jayakumaran Nair, Sabulal Baby

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Original Research

Evaluation of homodimer 99mTc-HYNIC-E(SSSLTVPWY)2 peptide on HER2-over expressed breast cancer cells

Fatemeh Ebrahimi, Zohreh Noaparast, Seyed Jalal Hosseinimehr

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Original Research

In silico and in vitro studies of novel cyanoacrylamides incorporating pyrazole moiety against breast and prostate carcinomas

Farid M. Sroor, Karima F. Mahrous, Heba I. Shafey, Nedal R. Eid, Ismail A. Abdelhamid, Nada S. Ibrahim

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Faridoon .

Senior Synthetic Medicinal Chemist I Project Manager at Drug Design and Development Center, Suzhou Genhouse Pharmaceutical Co., Ltd.

1 年

Nice to see our work featured on the cover page of Medicinal Chemistry Research.

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