Dr. GPCR

New course alert ?? The next Dr. GPCR course on the Development of GPCR Ligands as Therapeutic Drugs, is open for registration. The course will cover: The Essentials of New Drug Development Drug Clearance; the Engine of Pharmacokinetics Whole Body Pharmacokinetics and Therapeutic Profiles Essential Early Drug Safety Be the first to register, save your spot, spread the word, and enjoy a 25% discount with your Premium Membership ?? Go to https://lnkd.in/d5_fWVNH for more information! #gpcr #drgpcr #drugdiscovery #biotech #drugsafety Andreína Martín Monserrat Avila-Zozaya Mark Schmeizl Sam Hoare Cam Sinh Lu John Teye Azietaku, PhD Shivani Sachdev, PhD Terry Hebert Terry Kenakin Brian Arey

How does nanoscale GPCR organization shape signaling? ?? We explore this & more with Dr. Gabriele Kockelkoren, a physicist-turned-biologist with expertise in GPCR spatial dynamics. And if you wonder what his favorite GPCR could be, here’s the answer ?? ? Listen now https://lnkd.in/eZjhkRmn #gpcr #drgpcr

?? Why Does GPCR Location Make All the Difference? GPCR location within the cell can change everything: function, pharmacology, and even drug response. In Ep.162 of the Dr.GPCR Podcast, Dr. Gabriele Kockelkoren dives into: ?? How GPCR trafficking shapes signaling outcomes ?? Career insights from the lab to the broader biotech world This episode is packed with knowledge for scientists, drug hunters, and anyone fascinated by GPCRs! ??? Listen now https://lnkd.in/eZjhkRmn #DrGPCR #GPCR #DrugDiscovery #Pharma #Biotech #SciencePodcast ? Tune in today!

?? Are Your GPCR Bioassays Telling the Whole Story? Modifying signaling proteins in bioassays can be a double-edged sword—enhancing detection but also distorting reality. How do we balance sensitivity with biological relevance? In our latest article, we dive into: ?? The risks of altering GPCR signaling proteins ??? Best practices to keep your assays biologically meaningful ?? How to design better experiments without misleading results Read Dr Kiyan Afzali's article today: https://lnkd.in/eFuXv-27 #GPCR #DrugDiscovery #Bioassays #Pharmacology #LabScience

Do you remember the first time you were left alone in the lab with an experiment? ?? Did your experience compare to Dr. Brian Hudson’s? ?? Tune into this week’s Dr. GPCR Podcast for great stories, GPCR insights, and a fascinating journey that led Dr. Hudson to years of groundbreaking research at the University of Glasgow. Don’t miss out! ?Listen now https://lnkd.in/eyv_NyVB #gpcr #drgpcr

A large-scale analysis of GPCR molecular dynamics reveals hidden allosteric sites and lateral gateways, unlocking new possibilities for drug discovery. Subscribe to the Dr. GPCR Newsletter ?? and get the latest GPCR News delivered to your inbox ??https://lnkd.in/ewjYimXh #gpcr#drgpcr

?? Final Call! Don’t miss Dr. Terry Kenakin’s expert-led course on GPCR drug development—learn from one of the best in the field! ?? Are You Keeping Up with the Fast-Paced World of GPCR Drug Discovery? GPCRs remain one of the most critical target classes in drug development, yet new discoveries and technologies constantly reshape the field. Here’s what’s making waves this week: ?? GPR88’s Role in Kappa Opioid Receptor Signaling – Unlocking new insights into GPCR modulation and potential therapeutic applications. ?? AI-Powered GPCR Drug Screening – How machine learning is accelerating hit discovery and lead optimization for complex GPCR targets. ?? Stay ahead with the latest GPCR research and industry trends: https://lnkd.in/e8giSFAf #GPCR #DrGPCR #Science #DrugDiscovery #Pharma #Biotech #GProteinCoupledReceptors #GPCRresearch

Ep.161 of the Dr. GPCR Podcast is here! ?? Join us as we chat with Dr. Brian Hudson about the scientist’s journey—his learnings, lab experiences, and the unexpected paths GPCRs can take you on! ?? ?An episode you can’t miss https://lnkd.in/eyv_NyVB #gpcr #drgpcr

?? Exciting Opportunity for Professionals in Drug Development! ?? Register today for a one-of-a-kind online course at Dr. GPCR University: "Development of GPCR Ligands as Therapeutic Drugs." ?? Dates: March 20 - April 10, 2025 ? Time: Thursdays, 10:00 AM - 11:30 AM (EST) This advanced course is essential for anyone working in drug development and focuses on: The essentials of new drug development Key pharmacokinetic elements (absorption, distribution, clearance) Hepatic metabolism and the Cytochrome P450 system Drug safety and toxicology (including drug-drug interactions) And much more! Gain deep insights into GPCR drug candidates and learn the critical assays and techniques required to bring therapeutic molecules to life. ?? Only 25 spots available — register now! ?? This is a great opportunity for both academia and industry professionals. Sessions will be live, and you’ll also have 1:1 discussion time with the instructor. Full PDFs of the slides will be available! ?? https://lnkd.in/d5_fWVNH #GPCR #DrugDevelopment #Pharmacokinetics #TherapeuticDrugs #OnlineCourse #DrGPCRUniversity #PharmaceuticalIndustry

?? Enhance Your GPCR Expertise with Dr. GPCR University! Looking to sharpen your skills in GPCR pharmacology, drug discovery, data analysis, or project management? Dr.GPCR University offers industry-focused courses designed to help you stay ahead in the field. ? Comprehensive course library covering cutting-edge GPCR science ? Practical insights for real-world drug discovery challenges ? Flexible, on-demand learning to fit your schedule ?? Elevate your expertise today: Start learning now #GPCR #Pharmacology #DrugDiscovery #Biotech #DrGPCR